Name | N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl-2-pyrrolidinedicarboxamide |
Synonyms | TCS-102 TCS 1102 N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl-2-pyrrolidinedicarboxamide (2S)-N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl]-2-pyrrolidinecarboxamide (2S)- 2-Pyrrolidinecarboxamide, N-[1,1'-biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl] 2-PyrrolidinecarboxaMide, N-[1,1'-biphenyl]-2-yl-1-[2-[(1-Methyl-1H-benziMidazol-2-yl)thio]acetyl]-, (2S)- (2S)-N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl]-2-pyrrolidinecarboxamide TCS1102 TCS 1102 N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl-2-pyrrolidinedicarboxamide |
CAS | 916141-36-1 |
Molecular Formula | C27H26N4O2S |
Molar Mass | 470.59 |
Storage Condition | Sealed in dry,2-8°C |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 2.125 ml | 10.625 ml | 21.25 ml |
5 mM | 0.425 ml | 2.125 ml | 4.25 ml |
10 mM | 0.213 ml | 1.063 ml | 2.125 ml |
5 mM | 0.043 ml | 0.213 ml | 0.425 ml |
biological activity | TCS 1102 is an orexin OX receptor antagonist, and Ki for OX2 and OX1 receptors are 0.2 and 3 nM respectively. |